SGC0946 is a highly potent and selective DOT1L methyltransferase inhibitor with IC50 of 0.3 nM; selectively kill mixed lineage leukaemia cells.
Target
DOT1L
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IC50 Value
0.3nM
Diseases and Conditions
Cancer
体外
体内
Chemical information:
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分子量
618.57
储存条件
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3 years -20 ℃ powder
2 years -80 ℃ In solvent
分子式
C28H40BrN7O4
CAS:
1561178-17-3
备注
For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.
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溶解度
体外
Ethanol
100mg/mL(161.66mM)
DMSO
100mg/ml(161.66 mM)
Water
<1mg/ml
体内
* <1 mg/ml refers to the product slightly soluble or insoluble